Flumazenil is an imidazo-benzodiazepine derivative, effective in reversing benzodiazepine-induced activities and available by injection and intranasal.
It has antagonistic and antidote properties to therapeutically used benzodiazepines, through competitive inhibition
Product Name |
Flumazenil |
CAS Number |
78755-81-4 |
Therapeutic Class |
Antidote, Anesthesia reversal, Reversal of sedation caused by benzodiazepine |
Dosage Form |
Solution for Injection |
Availability |
Commercial |
Regulatory Status |
USDMF, CEP, JDMF, KDMF, CADMF |